Kulkarni, Ashish A.; Roy, Bhaskar; Rao, Poornima S.; Wyant, Gregory A.; Mahmoud, Ayaat; Ramachandran, Madhumitha; Sengupta, Poulomi; Goldman, Aaron; Kotamraju, Venkata Ramana; BASU, SUDIPTA; Mashelkar, Raghunath A.; Ruoslahti, Erkki; Dinulescu, Daniela M.; Sengupta, Shiladitya
(American Association for Cancer Research, 2013-12)
The centrality of phosphoinositide-3-kinase (PI3K) in cancer etiology is well established, but clinical translation of PI3K inhibitors has been limited by feedback signaling, suboptimal intratumoral concentration, and an ...